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-Structure paper
Title | Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 5391-5402, Year 2016 |
Publish date | Jan 9, 2016 (structure data deposition date) |
![]() | Crawford, T.D. / Tsui, V. / Flynn, E.M. / Wang, S. / Taylor, A.M. / Cote, A. / Audia, J.E. / Beresini, M.H. / Burdick, D.J. / Cummings, R. ...Crawford, T.D. / Tsui, V. / Flynn, E.M. / Wang, S. / Taylor, A.M. / Cote, A. / Audia, J.E. / Beresini, M.H. / Burdick, D.J. / Cummings, R. / Dakin, L.A. / Duplessis, M. / Good, A.C. / Hewitt, M.C. / Huang, H.R. / Jayaram, H. / Kiefer, J.R. / Jiang, Y. / Murray, J. / Nasveschuk, C.G. / Pardo, E. / Poy, F. / Romero, F.A. / Tang, Y. / Wang, J. / Xu, Z. / Zawadzke, L.E. / Zhu, X. / Albrecht, B.K. / Magnuson, S.R. / Bellon, S. / Cochran, A.G. |
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Methods | X-ray diffraction |
Resolution | 1.0402 - 1.5 Å |
Structure data | ![]() PDB-5i1q: ![]() PDB-5i29: ![]() PDB-5i40: ![]() PDB-5i7x: ![]() PDB-5i7y: ![]() PDB-5i80: ![]() PDB-5i88: |
Chemicals | ![]() ChemComp-67C: ![]() ChemComp-HOH: ![]() ChemComp-67B: ![]() ChemComp-CA: ![]() ChemComp-EDO: ![]() ChemComp-PEG: ![]() ChemComp-67N: ![]() ChemComp-69G: ![]() ChemComp-DMS: ![]() ChemComp-PGE: ![]() ChemComp-GOL: |
Source |
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![]() | PROTEIN BINDING/INHIBITOR / TAF1(2) Second Bromodomain of TAF1 Small-molecule ligand bound / PROTEIN BINDING-INHIBITOR complex / TAF1(2) / second bromodomain of TAF1 / inhibitor-bound / RNA BINDING PROTEIN / Bromodomain Inhibitor Epigenetics Structure-based drug design / TRANSCRIPTION / BRD9 / bromodomain / epigenetics / structure-based design / BRD4 / Structure-based drug design |