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-Structure paper
Title | Dissecting Therapeutic Resistance to ERK Inhibition. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 15, Page 548-559, Year 2016 |
Publish date | Jan 4, 2016 (structure data deposition date) |
![]() | Jha, S. / Morris, E.J. / Hruza, A. / Mansueto, M.S. / Schroeder, G.K. / Arbanas, J. / McMasters, D. / Restaino, C.R. / Dayananth, P. / Black, S. ...Jha, S. / Morris, E.J. / Hruza, A. / Mansueto, M.S. / Schroeder, G.K. / Arbanas, J. / McMasters, D. / Restaino, C.R. / Dayananth, P. / Black, S. / Elsen, N.L. / Mannarino, A. / Cooper, A. / Fawell, S. / Zawel, L. / Jayaraman, L. / Samatar, A.A. |
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Methods | X-ray diffraction |
Resolution | 1.45 - 1.69 Å |
Structure data | ![]() PDB-5hd4: ![]() PDB-5hd7: |
Chemicals | ![]() ChemComp-38Z: ![]() ChemComp-SO4: ![]() ChemComp-PG4: ![]() ChemComp-DMS: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE / SERINE/THREONINE-PROTEIN KINASE / MAP KINASE / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX |