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-Structure paper
Title | Potent and Selective Bivalent Inhibitors of Bet Bromodomains |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 12, Page 1097-, Year 2016 |
Publish date | Aug 19, 2015 (structure data deposition date) |
Authors | Waring, M.J. / Chen, H. / Rabow, A.A. / Walker, G. / Bobby, R. / Boiko, S. / Bradbury, R.H. / Callis, R. / Clark, E. / Dale, I. ...Waring, M.J. / Chen, H. / Rabow, A.A. / Walker, G. / Bobby, R. / Boiko, S. / Bradbury, R.H. / Callis, R. / Clark, E. / Dale, I. / Daniels, D.L. / Dulak, A. / Flavell, L. / Holdgate, G. / Jowitt, T.A. / Kikhney, A. / Mcalister, M. / Ogg, D. / Patel, J. / Petteruti, P. / Robb, G.R. / Robers, M.B. / Saif, S. / Stratton, N. / Svergun, D.I. / Wang, W. / Whittaker, D. / Wilson, D.M. / Yao, Y. |
External links | Nat. Chem. Biol. / PubMed:27775716 |
Methods | X-ray diffraction |
Resolution | 1.49 - 2.01 Å |
Structure data | PDB-5ad2: PDB-5ad3: |
Chemicals | ChemComp-ETU: ChemComp-HOH: ChemComp-K6K: |
Source |
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Keywords | TRANSCRIPTION |