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-Structure paper
Title | Structure-Based Design of GNE-495, a Potent and Selective MAP4K4 Inhibitor with Efficacy in Retinal Angiogenesis. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 913-918, Year 2015 |
Publish date | Apr 29, 2015 (structure data deposition date) |
![]() | Ndubaku, C.O. / Crawford, T.D. / Chen, H. / Boggs, J.W. / Drobnick, J. / Harris, S.F. / Jesudason, R. / McNamara, E. / Nonomiya, J. / Sambrone, A. ...Ndubaku, C.O. / Crawford, T.D. / Chen, H. / Boggs, J.W. / Drobnick, J. / Harris, S.F. / Jesudason, R. / McNamara, E. / Nonomiya, J. / Sambrone, A. / Schmidt, S. / Smyczek, T. / Vitorino, P. / Wang, L. / Wu, P. / Yeung, S. / Chen, J. / Chen, K. / Ding, C.Z. / Wang, T. / Xu, Z. / Gould, S.E. / Murray, L.J. / Ye, W. |
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Methods | X-ray diffraction |
Resolution | 2.89 Å |
Structure data | ![]() PDB-4zk5: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-MES: ![]() ChemComp-4P4: ![]() ChemComp-HOH: |
Source |
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![]() | Transferase/Transferase Inhibitor / kinase / Transferase-Transferase Inhibitor complex |