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-Structure paper
Title | Pyridopyrimidinone Derivatives as Potent and Selective c-Jun N-Terminal Kinase (JNK) Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 413-418, Year 2015 |
Publish date | Feb 10, 2015 (structure data deposition date) |
![]() | Zheng, K. / Park, C.M. / Iqbal, S. / Hernandez, P. / Park, H. / LoGrasso, P.V. / Feng, Y. |
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Methods | X-ray diffraction |
Resolution | 2.04 - 2.055 Å |
Structure data | ![]() PDB-4y46: ![]() PDB-4y5h: |
Chemicals | ![]() ChemComp-4F2: ![]() ChemComp-HOH: ![]() ChemComp-519: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / JNK / MAP kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex |