+Search query
-Structure paper
Title | Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 Tool Compound. |
---|---|
Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 655-659, Year 2015 |
Publish date | Feb 9, 2015 (structure data deposition date) |
Authors | Mitchell, L.H. / Drew, A.E. / Ribich, S.A. / Rioux, N. / Swinger, K.K. / Jacques, S.L. / Lingaraj, T. / Boriack-Sjodin, P.A. / Waters, N.J. / Wigle, T.J. ...Mitchell, L.H. / Drew, A.E. / Ribich, S.A. / Rioux, N. / Swinger, K.K. / Jacques, S.L. / Lingaraj, T. / Boriack-Sjodin, P.A. / Waters, N.J. / Wigle, T.J. / Moradei, O. / Jin, L. / Riera, T. / Porter-Scott, M. / Moyer, M.P. / Smith, J.J. / Chesworth, R. / Copeland, R.A. |
External links | Acs Med. Chem. Lett. / PubMed:26101569 |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.37 Å |
Structure data | PDB-4y2h: PDB-4y30: |
Chemicals | ChemComp-SAH: ChemComp-49K: ChemComp-GOL: ChemComp-HOH: ChemComp-49L: ChemComp-MG: |
Source |
|
Keywords | TRANSFERASE |