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-Structure paper
Title | Structure-Based Design of Type II Inhibitors Applied to Maternal Embryonic Leucine Zipper Kinase. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 6, Page 31-, Year 2015 |
Publish date | May 21, 2014 (structure data deposition date) |
Authors | Johnson, C.N. / Adelinet, C. / Berdini, V. / Beke, L. / Bonnet, P. / Brehmer, D. / Calo, F. / Coyle, J.E. / Day, P.J. / Frederickson, M. ...Johnson, C.N. / Adelinet, C. / Berdini, V. / Beke, L. / Bonnet, P. / Brehmer, D. / Calo, F. / Coyle, J.E. / Day, P.J. / Frederickson, M. / Freyne, E.J.E. / Gilissen, R.A.H.J. / Hamlett, C.C.F. / Howard, S. / Meerpoel, L. / Mevellec, L. / Mcmenamin, R. / Pasquier, E. / Patel, S. / Rees, D.C. / Linders, J.T.M. |
External links | Acs Med. Chem. Lett. / PubMed:25589926 |
Methods | X-ray diffraction |
Resolution | 1.98 - 2.02 Å |
Structure data | PDB-4umt: PDB-4umu: |
Chemicals | ChemComp-DMS: ChemComp-47W: ChemComp-HOH: ChemComp-0V0: |
Source |
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Keywords | TRANSFERASE / FRAGMENT BASED DRUG DESIGN / KINASE |