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Title | Back Pocket Flexibility Provides Group II p21-Activated Kinase (PAK) Selectivity for Type I 1/2 Kinase Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 57, Page 1033-1045, Year 2014 |
Publish date | Dec 14, 2013 (structure data deposition date) |
![]() | Staben, S.T. / Feng, J.A. / Lyle, K. / Belvin, M. / Boggs, J. / Burch, J.D. / Chua, C.C. / Cui, H. / Dipasquale, A.G. / Friedman, L.S. ...Staben, S.T. / Feng, J.A. / Lyle, K. / Belvin, M. / Boggs, J. / Burch, J.D. / Chua, C.C. / Cui, H. / Dipasquale, A.G. / Friedman, L.S. / Heise, C. / Koeppen, H. / Kotey, A. / Mintzer, R. / Oh, A. / Roberts, D.A. / Rouge, L. / Rudolph, J. / Tam, C. / Wang, W. / Xiao, Y. / Young, A. / Zhang, Y. / Hoeflich, K.P. |
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Methods | X-ray diffraction |
Resolution | 2.2 - 2.8 Å |
Structure data | ![]() PDB-4o0r: ![]() PDB-4o0t: ![]() PDB-4o0v: ![]() PDB-4o0x: ![]() PDB-4o0y: |
Chemicals | ![]() ChemComp-7KC: ![]() ChemComp-HOH: ![]() ChemComp-2OL: ![]() ChemComp-2OQ: ![]() ChemComp-2OO: |
Source |
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![]() | transferase/transferase inhibitor / PAK1 / transferase-transferase inhibitor complex / PAK4 |