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-Structure paper
Title | Targeting low-druggability bromodomains: fragment based screening and inhibitor design against the BAZ2B bromodomain. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 10183-10187, Year 2013 |
Publish date | Nov 26, 2013 (structure data deposition date) |
Authors | Ferguson, F.M. / Fedorov, O. / Chaikuad, A. / Philpott, M. / Muniz, J.R. / Felletar, I. / von Delft, F. / Heightman, T. / Knapp, S. / Abell, C. / Ciulli, A. |
External links | J. Med. Chem. / PubMed:24304323 |
Methods | X-ray diffraction |
Resolution | 1.85 - 2.08 Å |
Structure data | PDB-4nr9: PDB-4nra: PDB-4nrb: PDB-4nrc: |
Chemicals | ChemComp-EDO: ChemComp-ALY: ChemComp-HOH: ChemComp-2LW: ChemComp-2LX: ChemComp-2LY: ChemComp-15P: |
Source |
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Keywords | TRANSCRIPTION / SGC / Structural Genomics Consortium / bromodomain / acetylated lysine binding protein / KIAA1476 / WALp4 |