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-Structure paper
Title | Replacement of Water Molecules in a Phosphate Binding Site by Furanoside-Appended lin-Benzoguanine Ligands of tRNA-Guanine Transglycosylase (TGT). |
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Journal, issue, pages | Chemistry, Vol. 21, Page 126-135, Year 2015 |
Publish date | May 24, 2013 (structure data deposition date) |
Authors | Barandun, L.J. / Ehrmann, F.R. / Zimmerli, D. / Immekus, F. / Giroud, M. / Grunenfelder, C. / Schweizer, W.B. / Bernet, B. / Betz, M. / Heine, A. ...Barandun, L.J. / Ehrmann, F.R. / Zimmerli, D. / Immekus, F. / Giroud, M. / Grunenfelder, C. / Schweizer, W.B. / Bernet, B. / Betz, M. / Heine, A. / Klebe, G. / Diederich, F. |
External links | Chemistry / PubMed:25483606 |
Methods | X-ray diffraction |
Resolution | 1.17 - 1.405 Å |
Structure data | PDB-4kwo: PDB-4lbu: PDB-4leq: |
Chemicals | ChemComp-1UD: ChemComp-ZN: ChemComp-GOL: ChemComp-HOH: ChemComp-1WJ: ChemComp-CL: ChemComp-1WK: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE FURANOSIDE-BASED INHIBITOR COMPLEX / Tim Barrel / GLYCOSYLTRANSFERASE / Zinc-BINDING / TRANSFERASE-TRANSFERASE INHIBITOR complex / TRANSFERASE |