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-Structure paper
Title | Development of cyclic peptomer inhibitors targeting the polo-box domain of polo-like kinase 1. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 21, Page 2623-2634, Year 2013 |
Publish date | Sep 26, 2012 (structure data deposition date) |
Authors | Murugan, R.N. / Park, J.E. / Lim, D. / Ahn, M. / Cheong, C. / Kwon, T. / Nam, K.Y. / Choi, S.H. / Kim, B.Y. / Yoon, D.Y. ...Murugan, R.N. / Park, J.E. / Lim, D. / Ahn, M. / Cheong, C. / Kwon, T. / Nam, K.Y. / Choi, S.H. / Kim, B.Y. / Yoon, D.Y. / Yaffe, M.B. / Yu, D.Y. / Lee, K.S. / Bang, J.K. |
External links | Bioorg. Med. Chem. / PubMed:23498919 |
Methods | X-ray diffraction |
Resolution | 2 - 2.65 Å |
Structure data | PDB-4hab: PDB-4hy2: |
Chemicals | ChemComp-CXS: ChemComp-PO4: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Polo-box domain / PHOSPHOPROTEIN-BINDING DOMAIN / TRANSFERASE-TRANSFERASE INHIBITOR complex / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |