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-Structure paper
Title | Rational design of highly selective spleen tyrosine kinase inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 55, Page 10414-10423, Year 2012 |
Publish date | Jul 5, 2012 (structure data deposition date) |
Authors | Lucas, M.C. / Goldstein, D.M. / Hermann, J.C. / Kuglstatter, A. / Liu, W. / Luk, K.C. / Padilla, F. / Slade, M. / Villasenor, A.G. / Wanner, J. ...Lucas, M.C. / Goldstein, D.M. / Hermann, J.C. / Kuglstatter, A. / Liu, W. / Luk, K.C. / Padilla, F. / Slade, M. / Villasenor, A.G. / Wanner, J. / Xie, W. / Zhang, X. / Liao, C. |
External links | J. Med. Chem. / PubMed:23151054 |
Methods | X-ray diffraction |
Resolution | 1.4 - 2.318 Å |
Structure data | PDB-4fyn: PDB-4fyo: PDB-4fz6: |
Chemicals | ChemComp-0VE: ChemComp-HOH: ChemComp-0VF: ChemComp-0VG: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / kinase inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |