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-Structure paper
Title | Development of Novel In Vivo Chemical Probes to Address CNS Protein Kinase Involvement in Synaptic Dysfunction. |
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Journal, issue, pages | Plos One, Vol. 8, Page e66226-e66226, Year 2013 |
Publish date | May 21, 2012 (structure data deposition date) |
![]() | Watterson, D.M. / Grum-Tokars, V.L. / Roy, S.M. / Schavocky, J.P. / Bradaric, B.D. / Bachstetter, A.D. / Xing, B. / Dimayuga, E. / Saeed, F. / Zhang, H. ...Watterson, D.M. / Grum-Tokars, V.L. / Roy, S.M. / Schavocky, J.P. / Bradaric, B.D. / Bachstetter, A.D. / Xing, B. / Dimayuga, E. / Saeed, F. / Zhang, H. / Staniszewski, A. / Pelletier, J.C. / Minasov, G. / Anderson, W.F. / Arancio, O. / Van Eldik, L.J. |
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Methods | X-ray diffraction |
Resolution | 1.85 - 2 Å |
Structure data | ![]() PDB-4f9w: ![]() PDB-4f9y: ![]() PDB-4fa2: |
Chemicals | ![]() ChemComp-GG5: ![]() ChemComp-LM4: ![]() ChemComp-ZN: ![]() ChemComp-ACT: ![]() ChemComp-BME: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-LM3: ![]() ChemComp-PEG: ![]() ChemComp-SB0: ![]() ChemComp-EDO: |
Source |
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![]() | transferase/transferase inhibitor / protein kinase catalytic domain / transferase-transferase inhibitor complex |