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-Structure paper
Title | Antidotes to anthrax lethal factor intoxication. Part 3: Evaluation of core structures and further modifications to the C2-side chain. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 22, Page 2242-, Year 2012 |
Publish date | Feb 22, 2012 (structure data deposition date) |
Authors | Jiao, G.S. / Kim, S. / Moayeri, M. / Crown, D. / Thai, A. / Cregar-Hernandez, L. / McKasson, L. / Sankaran, B. / Lehrer, A. / Wong, T. ...Jiao, G.S. / Kim, S. / Moayeri, M. / Crown, D. / Thai, A. / Cregar-Hernandez, L. / McKasson, L. / Sankaran, B. / Lehrer, A. / Wong, T. / Johns, L. / Margosiak, S.A. / Leppla, S.H. / Johnson, A.T. |
External links | Bioorg. Med. Chem. Lett. / PubMed:22342144 |
Methods | X-ray diffraction |
Resolution | 1.632 Å |
Structure data | PDB-4dv8: |
Chemicals | ChemComp-ZN: ChemComp-0LX: ChemComp-MLI: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / endopeptidase / Zinc dependent |