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-Structure paper
Title | The Structure Based Design of Dual Hdac/Bet Inhibitors as Novel Epigenetic Probes. |
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Journal, issue, pages | Medchemcomm, Vol. 5, Page 342-, Year 2014 |
Publish date | Jan 13, 2014 (structure data deposition date) |
Authors | Atkinson, S.J. / Soden, P.E. / Angell, D.C. / Bantscheff, M. / Chung, C. / Giblin, K.A. / Smithers, N. / Furze, R.C. / Gordon, L. / Drewes, G. ...Atkinson, S.J. / Soden, P.E. / Angell, D.C. / Bantscheff, M. / Chung, C. / Giblin, K.A. / Smithers, N. / Furze, R.C. / Gordon, L. / Drewes, G. / Rioja, I. / Witherington, J. / Parr, N.J. / Prinjha, R.K. |
External links | Medchemcomm / Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.4 - 1.6 Å |
Structure data | PDB-4cl9: PDB-4clb: |
Chemicals | ChemComp-EDO: ChemComp-IES: ChemComp-HOH: ChemComp-83T: |
Source |
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Keywords | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / ANTAGONIST |