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-Structure paper
Title | R-Configuration of 4-Aminopyridyl-Based Inhibitors of Cyp51 Confers Superior Efficacy Against Trypanosoma Cruzi |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 5, Page 434-, Year 2014 |
Publish date | Jul 16, 2013 (structure data deposition date) |
Authors | Choi, J.Y. / Calvet, C.M. / Vieira, D.F. / Gunatilleke, S.S. / Cameron, M.D. / Mckerrow, J.H. / Podust, L.M. / Roush, W.R. |
External links | Acs Med. Chem. Lett. / PubMed:24900854 |
Methods | X-ray diffraction |
Resolution | 3.1 Å |
Structure data | PDB-4by0: |
Chemicals | ChemComp-HEM: ChemComp-5PS: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE / STEROL 14-DEMETHYLASE / STEROL BIOSYNTHESIS / CHAGAS DISEASE |