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-Structure paper
Title | Discovery of a Potent and Isoform-Selective Targeted Covalent Inhibitor of the Lipid Kinase Pi3Kalpha |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 712-, Year 2013 |
Publish date | Jan 9, 2013 (structure data deposition date) |
Authors | Nacht, M. / Qiao, L. / Sheets, M.P. / Martin, T.S. / Labenski, M. / Mazdiyasni, H. / Karp, R. / Zhu, Z. / Chaturvedi, P. / Bhavsar, D. ...Nacht, M. / Qiao, L. / Sheets, M.P. / Martin, T.S. / Labenski, M. / Mazdiyasni, H. / Karp, R. / Zhu, Z. / Chaturvedi, P. / Bhavsar, D. / Niu, D. / Westlin, W. / Petter, R.C. / Medikonda, A.P. / Singh, J. |
External links | J. Med. Chem. / PubMed:23360348 |
Methods | X-ray diffraction |
Resolution | 2.85 Å |
Structure data | PDB-3zim: |
Chemicals | ChemComp-KKR: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE |