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-Structure paper
Title | Structural and Functional Analyses of the Second-Generation Integrase Strand Transfer Inhibitor Dolutegravir (S/GSK1349572). |
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Journal, issue, pages | Mol. Pharmacol., Vol. 80, Page 565-572, Year 2011 |
Publish date | May 18, 2011 (structure data deposition date) |
Authors | Hare, S. / Smith, S.J. / Metifiot, M. / Jaxa-Chamiec, A. / Pommier, Y. / Hughes, S.H. / Cherepanov, P. |
External links | Mol. Pharmacol. / PubMed:21719464 |
Methods | X-ray diffraction |
Resolution | 2.49 - 2.55 Å |
Structure data | PDB-3s3m: PDB-3s3n: PDB-3s3o: |
Chemicals | ChemComp-ZN: ChemComp-SO4: ChemComp-GOL: ChemComp-NH4: ChemComp-MG: ChemComp-DLU: ChemComp-HEZ: ChemComp-HOH: |
Source |
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Keywords | RECOMBINATION/INHIBITOR/DNA / PROTEIN-DNA COMPLEX / TETRAMER / DNA INTEGRATION / ENDONUCLEASE / METAL-BINDING / MULTIFUNCTIONAL ENZYME / NUCLEASE / NUCLEOTIDYLTRANSFERASE / NUCLEUS / TRANSFERASE / VIRAL NUCLEOPROTEIN / VIRION / DNA-BINDING / ZINC BINDING / HHCC MOTIF / VIRAL PROTEIN / RECOMBINATION / INHIBITOR / RECOMBINATION-INHIBITOR-DNA complex / TRANSFERASE/INHIBITOR/DNA / TRANSFERASE-INHIBITOR-DNA complex |