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-Structure paper
Title | Suppression of inflammation by a synthetic histone mimic |
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Journal, issue, pages | Nature, Vol. 468, Page 1119-1123, Year 2010 |
Publish date | Oct 9, 2010 (structure data deposition date) |
![]() | Nicodeme, E. / Jeffrey, K.L. / Schaefer, U. / Beinke, S. / Dewell, S. / Chung, C. / Chandwani, R. / Marazzi, I. / Wilson, P. / Coste, H. ...Nicodeme, E. / Jeffrey, K.L. / Schaefer, U. / Beinke, S. / Dewell, S. / Chung, C. / Chandwani, R. / Marazzi, I. / Wilson, P. / Coste, H. / White, J. / Kirilovsky, J. / Rice, C.M. / Lora, J.M. / Prinjha, R.K. / Lee, K. / Tarakhovsky, A. |
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Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | ![]() PDB-3p5o: |
Chemicals | ![]() ChemComp-EAM: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN/INHIBITOR / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / ANTAGONIST / IBET / inhibition of acetylated lysine histone binding / Transcription Regulator / SIGNALING PROTEIN-INHIBITOR complex |