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-Structure paper
Title | Conserved Binding Mode of Human beta(2) Adrenergic Receptor Inverse Agonists and Antagonist Revealed by X-ray Crystallography |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 132, Page 11443-11445, Year 2010 |
Publish date | Jul 14, 2010 (structure data deposition date) |
![]() | Wacker, D. / Fenalti, G. / Brown, M.A. / Katritch, V. / Abagyan, R. / Cherezov, V. / Stevens, R.C. |
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Methods | X-ray diffraction |
Resolution | 2.84 - 3.16 Å |
Structure data | ![]() PDB-3ny8: ![]() PDB-3ny9: ![]() PDB-3nya: |
Chemicals | ![]() ChemComp-CLR: ![]() ChemComp-JRZ: ![]() ChemComp-OLA: ![]() ChemComp-OLC: ![]() ChemComp-PGE: ![]() ChemComp-HOH: ![]() ChemComp-JSZ: ![]() ChemComp-JTZ: |
Source |
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![]() | MEMBRANE PROTEIN / G Protein-coupled receptor / Lysozyme / Fusion / Transducer / Adrenergic / G-Proteins / Arrestins / Adrenalin / ICI 118 / 551 / Glycosylation / Palmitoylation / Phosphorylation / HYDROLASE / Structural Genomics / PSI-2 / Protein Structure Initiative / Accelerated Technologies Center for Gene to 3D Structure / ATCG3D / GPCR Network / GPCR / Compound 2 / Adrenaline / Alprenolol / PSI-Biology |