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-Structure paper
Title | Insight into Binding of Phosphodiesterase-9A Selective Inhibitors by Crystal Structures and Mutagenesis |
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Journal, issue, pages | J. Med. Chem., Vol. 53, Page 1726-1731, Year 2010 |
Publish date | Oct 2, 2009 (structure data deposition date) |
![]() | Wang, H. / Luo, X. / Ye, M. / Hou, J. / Robinson, H. / Ke, H. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.5 - 2.7 Å |
Structure data | ![]() PDB-3k3e: ![]() PDB-3k3h: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-MG: ![]() ChemComp-PDB: ![]() ChemComp-HOH: ![]() ChemComp-BYE: |
Source |
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![]() | HYDROLASE / PDE9 / catalytic domain / cGMP / Manganese / Metal-binding / Phosphoprotein |