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Title | 1.45 A resolution crystal structure of recombinant PNP in complex with a pM multisubstrate analogue inhibitor bearing one feature of the postulated transition state. |
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Journal, issue, pages | Biochem. Biophys. Res. Commun., Vol. 391, Page 703-708, Year 2010 |
Publish date | Jan 14, 2009 (structure data deposition date) |
Authors | Chojnowski, G. / Breer, K. / Narczyk, M. / Wielgus-Kutrowska, B. / Czapinska, H. / Hashimoto, M. / Hikishima, S. / Yokomatsu, T. / Bochtler, M. / Girstun, A. ...Chojnowski, G. / Breer, K. / Narczyk, M. / Wielgus-Kutrowska, B. / Czapinska, H. / Hashimoto, M. / Hikishima, S. / Yokomatsu, T. / Bochtler, M. / Girstun, A. / Staron, K. / Bzowska, A. |
External links | Biochem. Biophys. Res. Commun. / PubMed:19944078 |
Methods | X-ray diffraction |
Resolution | 1.45 Å |
Structure data | PDB-3fuc: |
Chemicals | ChemComp-9D9: ChemComp-MG: ChemComp-AZI: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / purine nucleoside phosphorylase / recombinant / glycosyltransferase / 9-deazaguanine / multisubstrate analogue inhibitors / nucleoside-binding / phosphate-binding / binding site / trimer |