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-Structure paper
Title | Structure-activity relationships and X-ray structures describing the selectivity of aminopyrazole inhibitors for c-Jun N-terminal kinase 3 (JNK3) over p38. |
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Journal, issue, pages | J. Biol. Chem., Vol. 284, Page 12853-12861, Year 2009 |
Publish date | Dec 10, 2008 (structure data deposition date) |
Authors | Kamenecka, T. / Habel, J. / Duckett, D. / Chen, W. / Ling, Y.Y. / Frackowiak, B. / Jiang, R. / Shin, Y. / Song, X. / LoGrasso, P. |
External links | J. Biol. Chem. / PubMed:19261605 |
Methods | X-ray diffraction |
Resolution | 2.2 - 2.28 Å |
Structure data | PDB-3fi2: PDB-3fi3: |
Chemicals | ChemComp-JK1: ChemComp-EDO: ChemComp-HOH: ChemComp-JK2: |
Source |
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Keywords | TRANSFERASE / JNK3 / protein-inhibitor complex / Alternative splicing / ATP-binding / Chromosomal rearrangement / Cytoplasm / Epilepsy / Kinase / Nucleotide-binding / Phosphoprotein / Serine/threonine-protein kinase |