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-Structure paper
Title | Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. |
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Journal, issue, pages | Acta Crystallogr. ,Sect. D, Vol. 67, Page 763-773, Year 2011 |
Publish date | Oct 3, 2006 (structure data deposition date) |
![]() | Kukimoto-Niino, M. / Tokmakov, A. / Terada, T. / Ohbayashi, N. / Fujimoto, T. / Gomi, S. / Shiromizu, I. / Kawamoto, M. / Matsusue, T. / Shirouzu, M. / Yokoyama, S. |
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Methods | X-ray diffraction |
Resolution | 1.86 - 2.54 Å |
Structure data | ![]() PDB-2e0a: ![]() PDB-2zdx: ![]() PDB-2zdy: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ANP: ![]() ChemComp-HOH: ![]() ChemComp-P4A: ![]() ChemComp-ADP: ![]() ChemComp-EPE: |
Source |
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![]() | TRANSFERASE / PDK4 / kinase / ATP-binding / Structural Genomics / NPPSFA / National Project on Protein Structural and Functional Analyses / RIKEN Structural Genomics/Proteomics Initiative / RSGI / INHIBITOR / Carbohydrate metabolism / Glucose metabolism / Mitochondrion / Phosphoprotein / Transit peptide / ADP |