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-Structure paper
Title | Relationship of Potency and Resilience to Drug Resistant Mutations for GW420867X Revealed by Crystal Structures of Inhibitor Complexes for Wild-Type, Leu100Ile, Lys101Glu, and Tyr188Cys Mutant HIV-1 Reverse Transcriptases. |
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Journal, issue, pages | J. Med. Chem., Vol. 50, Page 2301-2309, Year 2007 |
Publish date | Jan 30, 2007 (structure data deposition date) |
Authors | Ren, J. / Nichols, C.E. / Chamberlain, P.P. / Weaver, K.L. / Short, S.A. / Chan, J.H. / Kleim, J.P. / Stammers, D.K. |
External links | J. Med. Chem. / PubMed:17441703 |
Methods | X-ray diffraction |
Resolution | 2.3 - 2.9 Å |
Structure data | PDB-2opp: PDB-2opq: PDB-2opr: PDB-2ops: |
Chemicals | ChemComp-PO4: ChemComp-MG: ChemComp-HBQ: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / HIV-1 REVERSE TRANSCRIPTASE / AIDS / NNRTI / GW420867X / DRUG RESISTANCE |