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-Structure paper
Title | Structure-based design of a novel thiazolone scaffold as HCV NS5B polymerase allosteric inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 16, Page 5888-5891, Year 2006 |
Publish date | Aug 1, 2006 (structure data deposition date) |
Authors | Yan, S. / Appleby, T. / Larson, G. / Wu, J.Z. / Hamatake, R. / Hong, Z. / Yao, N. |
External links | Bioorg. Med. Chem. Lett. / PubMed:16934455 |
Methods | X-ray diffraction |
Resolution | 2 - 2.3 Å |
Structure data | PDB-2hwh: PDB-2hwi: |
Chemicals | ChemComp-RNA: ChemComp-HOH: ChemComp-VRX: |
Source |
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Keywords | TRANSFERASE / HCV / NS5B / Viral RNA-directed RNA Polymerase / RdRP / allosteric inhibitor / HCV inhibitor complex |