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-Structure paper
Title | Phenylethylthiazolylthiourea (PETT) non-nucleoside inhibitors of HIV-1 and HIV-2 reverse transcriptases. Structural and biochemical analyses. |
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Journal, issue, pages | J. Biol. Chem., Vol. 275, Page 5633-5639, Year 2000 |
Publish date | Jan 13, 2000 (structure data deposition date) |
![]() | Ren, J. / Diprose, J. / Warren, J. / Esnouf, R.M. / Bird, L.E. / Ikemizu, S. / Slater, M. / Milton, J. / Balzarini, J. / Stuart, D.I. / Stammers, D.K. |
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Methods | X-ray diffraction |
Resolution | 2.8 - 3 Å |
Structure data | ![]() PDB-1dtq: ![]() PDB-1dtt: |
Chemicals | ![]() ChemComp-FPT: ![]() ChemComp-HOH: ![]() ChemComp-FTC: |
Source |
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![]() | HYDROLASE/TRANSFERASE / HIV-1 reverse transcriptase AIDS / non-nucleoside inhibitor / drug design / HYDROLASE-TRANSFERASE COMPLEX |