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-Structure paper
Title | XChem fragment screen |
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Journal, issue, pages | To Be Published |
Publish date | Feb 28, 2020 (structure data deposition date) |
![]() | Talon, R. / Krojer, T. / Fairhead, M. / Sethi, R. / Bradley, A.R. / Aimon, A. / Collins, P. / Brandao-Neto, J. / Douangamath, A. / Wright, N. ...Talon, R. / Krojer, T. / Fairhead, M. / Sethi, R. / Bradley, A.R. / Aimon, A. / Collins, P. / Brandao-Neto, J. / Douangamath, A. / Wright, N. / MacLean, E. / Zhang, R. / Dias, A. / Brennan, P.E. / Bountra, C. / Arrowsmith, C.H. / Edwards, A. / von Delft, F. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.29 - 1.84 Å |
Structure data | ![]() PDB-5r4v: ![]() PDB-5r4w: ![]() PDB-5r4x: ![]() PDB-5r4y: ![]() PDB-5r4z: |
Chemicals | ![]() ChemComp-JMM: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-RWP: ![]() ChemComp-K3D: ![]() ChemComp-GX4: ![]() ChemComp-GWA: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / PanDDA / SGC - Diamond I04-1 fragment screening / XChemExplorer / ATPASE FAMILY / AAA DOMAIN CONTAINING 2 / ANCCA / AAA+ NUCLEAR COREGULATOR CANCER-ASSOCIATED PRO2000 PROTEIN / TWO AAA DOMAIN CONTAINING PROTEIN / SGC / STRUCTURAL GENOMICS CONSORTIUM / ATP-BINDING / BROMODOMAIN / NUCLEOTIDE-BINDING / PHOSPHOPROTEIN / SIGNALING PROTEIN / HYDROLASE-HYDROLASE INHIBITOR complex |