+Search query
-Structure paper
Title | Systematically Mitigating the p38alpha Activity of Triazole-based BET Inhibitors |
---|---|
Journal, issue, pages | ACS Med. Chem. Lett., Vol. 10, Page 1296-1301, Year 2019 |
Publish date | Mar 12, 2021 (structure data deposition date) |
![]() | Carlson, A.S. / Cui, H. / Divakaran, A. / Johnson, J.A. / Brunner, R.M. / Pomerantz, W.C.K. / Topczewski, J.J. |
![]() | ![]() |
Methods | X-ray diffraction |
Resolution | 1.42 Å |
Structure data | ![]() PDB-7m16: |
Chemicals | ![]() ChemComp-YNS: ![]() ChemComp-HOH: |
Source |
|
![]() | PROTEIN BINDING / inhibitor |