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-Structure paper
Title | Crystal structure and mechanistic analysis of a novel human kynurenine aminotransferase-2 reversible inhibitor |
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Journal, issue, pages | Med. Chem. Res., Year 2017 |
Publish date | Sep 24, 2016 (structure data deposition date) |
![]() | Nematollahi, A. / Sun, G. / Jayawickrama, G. / Hanrahan, J.R. / Church, W.B. |
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Methods | X-ray diffraction |
Resolution | 1.807 Å |
Structure data | ![]() PDB-5tf5: |
Chemicals | ![]() ChemComp-7AR: ![]() ChemComp-HOH: |
Source |
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![]() | transferase/transferase inhibitor / NS-1502 / reversible KAT-2 inhibitor / LLP / transferase-transferase inhibitor complex |