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| Title | Structural Determinants of the Binding and Activation of Estrogen Receptor alpha by Phenolic Thieno[2,3-d]pyrimidines |
|---|---|
| Journal, issue, pages | Helv. Chim. Acta, Vol. 106, Year 2023 |
| Publish date | Jul 29, 2021 (structure data deposition date) |
Authors | Reddy Sammeta, V. / Anderson, B.M. / Norris, J.D. / Torrice, C.D. / Joiner, C. / Liu, S. / Li, H. / Popov, K.I. / Fanning, S.W. / McDonnell, D.P. / Willson, T.M. |
External links | Helv. Chim. Acta / Search PubMed |
| Methods | X-ray diffraction |
| Resolution | 1.9 Å |
| Structure data | ![]() PDB-7rnm: |
| Chemicals | ![]() ChemComp-61Z: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSCRIPTION / Breast Cancer / Estrogen Receptor / Alpha Helical Bundle |
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