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-Structure paper
Title | Discovery of 2,6-disubstituted pyrazines as potent PI4K inhibitors with antimalarial activity |
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Journal, issue, pages | To Be Published |
Publish date | Apr 28, 2021 (structure data deposition date) |
![]() | Krake, S.H. / Martinez, P.D.G. / Poggi, M.L. / Ferreira, M.S. / Aguiar, A.C.C. / Souza, G.E. / Wenlock, M. / Jones, B. / Steinbrecher, T. / Day, T. ...Krake, S.H. / Martinez, P.D.G. / Poggi, M.L. / Ferreira, M.S. / Aguiar, A.C.C. / Souza, G.E. / Wenlock, M. / Jones, B. / Steinbrecher, T. / Day, T. / McPhail, J. / Burke, J. / Yeo, T. / Mok, S. / Uhlemann, A.C. / Fidock, D.A. / Chen, P. / Grodsky, N. / Deng, Y.L. / Guido, R.V.C. / Campbell, S.F. / Willis, P.A. / Dias, L.C. |
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Methods | X-ray diffraction |
Resolution | 2.91 Å |
Structure data | ![]() PDB-7mlk: |
Chemicals | ![]() ChemComp-ZHY: |
Source |
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![]() | TRANSFERASE/INHIBITOR / PI3K / pyrazine / complex / TRANSFERASE-INHIBITOR complex |