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-Structure paper
Title | 2-Aminothiazole-4-carboxylic acids as cross-class metallo-beta-lactamase inhibitors by mimicking beta-lactam hydrolysate binding |
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Journal, issue, pages | To Be Published |
Publish date | Jan 6, 2023 (structure data deposition date) |
![]() | Yan, Y.-H. / Zhu, K.-R. / Yang, L.-L. / Li, G.-B. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.151 - 2.193 Å |
Structure data | ![]() PDB-8hyb: ![]() PDB-8hyc: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-5ZX: ![]() ChemComp-ACT: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-60J: |
Source |
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![]() | HYDROLASE / Beta-lactamase class B IMP-1 / Beta-lactamase class B NDM-1 |