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Title | Small molecule AZD4635 inhibitor of A2AR signaling rescues immune cell function including CD103+ dendritic cells enhancing anti-tumor immunity |
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Journal, issue, pages | J Immunother Cancer, Year 2020 |
Publish date | Jun 15, 2018 (structure data deposition date) |
Authors | Borodovsky, A. / Barbon, C.M. / Wang, Y. / Ye, M. / Prickett, L. / Chandra, D. / Shaw, J. / Deng, N. / Sachsenmeier, K. / Clarke, J.D. ...Borodovsky, A. / Barbon, C.M. / Wang, Y. / Ye, M. / Prickett, L. / Chandra, D. / Shaw, J. / Deng, N. / Sachsenmeier, K. / Clarke, J.D. / Linghu, B. / Brown, G.A. / Brown, J. / Congreve, M. / Cheng, R.K.Y. / Dore, A.S. / Hurrell, E. / Shao, W. / Woessner, R. / Reimer, C. / Drew, L. / Fawell, S. / Schuller, A.G. / Mele, D.A. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | PDB-6gt3: |
Chemicals | ChemComp-NA: ChemComp-F9Q: ChemComp-CLR: ChemComp-OLA: ChemComp-OLC: ChemComp-HOH: |
Source |
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Keywords | MEMBRANE PROTEIN / 7TM / GPCR / SIGNALLING PROTEIN |