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Title | Novel Pure alphaVbeta3 Integrin Antagonists That Do Not Induce Receptor Extension, Prime the Receptor, or Enhance Angiogenesis at Low Concentrations |
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Journal, issue, pages | Acs Pharmacol Transl Sci, Vol. 2, Page 387-401, Year 2019 |
Publish date | Sep 24, 2018 (structure data deposition date) |
![]() | Li, J. / Fukase, Y. / Shang, Y. / Zou, W. / Munoz-Felix, J. / Buitrago, L. / van Agthoven, J. / Zhang, Y. / Hara, R. / Tanaka, Y. ...Li, J. / Fukase, Y. / Shang, Y. / Zou, W. / Munoz-Felix, J. / Buitrago, L. / van Agthoven, J. / Zhang, Y. / Hara, R. / Tanaka, Y. / Okamoto, R. / Yasui, T. / Nakahata, T. / Imaeda, T. / Aso, K. / Zhou, Y. / Locuson, C. / Nesic, D. / Duggan, M. / Takagi, J. / Vaughan, R.D. / Walz, T. / Hodivala-Dilke, K. / Teitelbaum, S.L. / Arnaout, M.A. / Filizola, M. / Foley, M.A. / Coller, B.S. |
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Methods | X-ray diffraction |
Resolution | 3.005 Å |
Structure data | ![]() PDB-6mk0: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-MN: ![]() ChemComp-JUY: ![]() ChemComp-HOH: |
Source |
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![]() | CELL ADHESION / HYBRID DOMAIN / PSI / EGF REPEATS / BETA TAIL / CALF / THIGH / BETA PROPELLER / RGD MOTIF / FIBRONECTIN / VITRONECTIN |