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-Structure paper
Title | Discovery of TAK-272: A Novel, Potent and Orally Active Renin Inhibitor |
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Journal, issue, pages | To be published |
Publish date | Jul 1, 2016 (structure data deposition date) |
![]() | Imaeda, Y. / Tokuhara, H. / Fukase, Y. / Kanagawa, R. / Kajimoto, Y. / Kusumoto, K. / Kondo, M. / Snell, G.P. / Behnke, C.A. / Kuroita, T. |
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Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | ![]() PDB-5kot: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-6VU: ![]() ChemComp-PGE: ![]() ChemComp-PEG: ![]() ChemComp-DMS: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE inhibitor / protein-inhibitor complex / HYDROLASE-HYDROLASE inhibitor complex |