+Search query
-Structure paper
Title | Targeting KAT6A/KAT6B dependencies in breast cancer with a novel selective, orally bioavailable KAT6 inhibitor, CTx-648/PF-9363 |
---|---|
Journal, issue, pages | To Be Published |
Publish date | Jun 17, 2022 (structure data deposition date) |
Authors | Sharma, S. / Chung, J. / Uryu, S. / Rickard, A. / Nady, N. / Cao, J. / Greasley, S.E. / Brodsky, O. / Khan, S. / Wang, H. ...Sharma, S. / Chung, J. / Uryu, S. / Rickard, A. / Nady, N. / Cao, J. / Greasley, S.E. / Brodsky, O. / Khan, S. / Wang, H. / Wang, Z. / Zhang, Y. / Tsaparikos, K. / Chen, L. / Mazurek, A. / Lapek, J. / Kung, P.P. / Sutton, S. / Richardson, P.A. / Greenwald, E. / Yamazaki, S. / Jones, R. / Maegley, K. / Bingham, P. / Lam, H. / Stupple, A.E. / Kamal, A. / Chueh, A. / Cuzzupe, A. / Morrow, B. / Ren, B. / Carrasco-Pozo, C. / Tan, T.W. / Bhuva, D. / Allan, E. / Surgenor, E. / Vaillant, F. / Pehlivanoglu, H. / Falk, H. / Whittle, J. / Newman, J.M. / Cursons, J. / Doherty, J.P. / White, K.L. / MacPherson, L. / Devlin, M. / Dennis, M.L. / Hattarki, M.K. / De Silva, M. / Camerino, M.A. / Butler, M.S. / Dolezal, O. / Pilling, P. / Foitzik, R. / Stupple, P.A. / Lagiakos, R. / Walker, S. / Hediyeh-Zadeh, S. / Nuttall, S. / Spall, S. / Charman, S.A. / Connor, T. / Peat, T.S. / Avery, V.M. / Bozikis, Y.E. / Yang, Y. / Zhang, M. / Monahan, B.J. / Voss, A.K. / Thomas, T. / Street, I.P. / Dawson, S.J. / Dawson, M. / Lindeman, G.J. / Davis, M. / Visvader, J.E. / Paul, T.A. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.58 Å |
Structure data | PDB-8dd5: |
Chemicals | ChemComp-R7L: ChemComp-ZN: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / histone lysine aceyltransferase / Inhibitor complex / Cancer / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |