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-Structure paper
Title | Crystal Structure of dual-specificity tyrosine phosphorylation regulated kinase 2 (DYRK2) in complex with an indirubin ligand |
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Journal, issue, pages | To be Published |
Publish date | Nov 30, 2009 (structure data deposition date) |
![]() | Filippakopoulos, P. / Myrianthopoulos, V. / Kritsanida, M. / Magiatis, P. / Skaltsounis, A.L. / Soundararajan, M. / Krojer, T. / Gileadi, O. / Hapka, E. / Fedorov, O. ...Filippakopoulos, P. / Myrianthopoulos, V. / Kritsanida, M. / Magiatis, P. / Skaltsounis, A.L. / Soundararajan, M. / Krojer, T. / Gileadi, O. / Hapka, E. / Fedorov, O. / Berridge, G. / Wang, J. / Shrestha, L. / Vollmar, M. / von Delft, F. / Arrowsmith, C.H. / Edwards, A. / Weigelt, J. / Bountra, C. / Mikros, E. / Knapp, S. |
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Methods | X-ray diffraction |
Resolution | 2.28 Å |
Structure data | ![]() PDB-3kvw: |
Chemicals | ![]() ChemComp-IRB: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / DYRK2 / dual-specificity tyrosine / ki-(Y)-phosphorylation regulated kinase 2 / PSK-H2 / kinase / Structural Genomics Consortium / SGC / Apoptosis / ATP-binding / Nucleotide-binding / Serine/threonine-protein kinase / Tyrosine-protein kinase |