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-Structure paper
Title | Crystal Structure of the Catalytic Domain of Human Jarid1B in Complex with 3D Fragment N,3-Dimethyl-N-(Pyridin-3-Ylmethyl)-1,2-Oxazole-5-Carboxamide (N10051A) (Ligand Modelled Based on Pandda Event Map, Sgc - Diamond I04-1 Fragment Screening) |
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Journal, issue, pages | To be Published |
Publish date | Mar 14, 2016 (structure data deposition date) |
Authors | Nowak, R. / Krojer, T. / Johansson, C. / Gileadi, C. / Kupinska, K. / Strain-Damerell, C. / Szykowska, A. / Talon, R. / Collins, P. / Burgess-Brown, N.A. ...Nowak, R. / Krojer, T. / Johansson, C. / Gileadi, C. / Kupinska, K. / Strain-Damerell, C. / Szykowska, A. / Talon, R. / Collins, P. / Burgess-Brown, N.A. / Arrowsmith, C.H. / Bountra, C. / Edwards, A.M. / von Delft, F. / Brennan, P.E. / Oppermann, U. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.05 Å |
Structure data | PDB-5fzk: |
Chemicals | ChemComp-ZN: ChemComp-CL: ChemComp-MN: ChemComp-EDO: ChemComp-NRW: ChemComp-PO4: ChemComp-DMS: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE / JARID1B / PLU1 / FRAGMENT SCREENING / STRUCTURAL GENOMICS CONSORTIUM / SGC / DIAMOND I04-1 / PANDDA |