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-Structure paper
Title | Discovery of TP0628103: A Selective MMP-7 Inhibitor Based on the Mitigation of OATP Substrate Recognition through Isoelectric Point Shift Strategy |
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Journal, issue, pages | To Be Published |
Publish date | Jul 20, 2023 (structure data deposition date) |
Authors | Oka, Y. / Abe-Sato, K. / Tabuse, H. / Yasukawa, Y. / Yahara, T. / Nishimoto, T. / Kamitani, M. / Fukunaga, T. / Ochiai, N. / Kumasaka-Abe, T. ...Oka, Y. / Abe-Sato, K. / Tabuse, H. / Yasukawa, Y. / Yahara, T. / Nishimoto, T. / Kamitani, M. / Fukunaga, T. / Ochiai, N. / Kumasaka-Abe, T. / Hitaka, K. / Gunji, E. / Ohara, H. / Takeda, T. / Kojima, N. / Asami, T. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.7 Å |
Structure data | PDB-8k4z: |
Chemicals | ChemComp-CA: ChemComp-ZN: ChemComp-IOD: ChemComp-CL: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / Matrilysin / Matrin / Matrix metalloproteinase-7 / Pump-1 protease / Uterine metalloproteinase |