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-Structure paper
Title | Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a Michael acceptor-based cyclic warhead scaffold |
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Journal, issue, pages | To Be Published |
Publish date | Jul 13, 2023 (structure data deposition date) |
Authors | Sok, P. / Poti, A. / Balint, D. / Soos, T. / Remenyi, A. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.65 - 2.55 Å |
Structure data | PDB-8psr: PDB-8pst: PDB-8psw: PDB-8psy: PDB-8pt0: PDB-8pt1: PDB-8pt3: PDB-8pt5: |
Chemicals | ChemComp-ANP: ChemComp-GOL: ChemComp-HOH: ChemComp-AN2:
ChemComp-DC6:
ChemComp-D2I:
ChemComp-EI0:
ChemComp-EAI:
ChemComp-E2A:
ChemComp-D7O:
ChemComp-D5R: |
Source |
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Keywords | SIGNALING PROTEIN / MAPK kinase / MAPK / inhibitor / covalent / ERK2 / Michael acceptor warhead |