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-Structure paper
Title | Discovery and in vivo evaluation of the potent and selective PI3K-delta inhibitors AM-0687 and AM-1430 |
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Journal, issue, pages | To Be Published |
Publish date | Jun 1, 2016 (structure data deposition date) |
Authors | Gonzalez-Lopez de Turiso, F. / Hao, X. / Shin, Y. / Bui, M. / Campuzano, I. / Cardozo, M. / Dunn, M.C. / Duquette, J. / Fisher, B. / Foti, R.S. ...Gonzalez-Lopez de Turiso, F. / Hao, X. / Shin, Y. / Bui, M. / Campuzano, I. / Cardozo, M. / Dunn, M.C. / Duquette, J. / Fisher, B. / Foti, R.S. / Henne, K. / He, X. / Hu, Y.-L. / Kelly, R.C. / Johnson, M.G. / Lucas, B.S. / McCarter, J. / McGee, L.R. / Medina, J.C. / Metz, D. / San Miguel, T. / Mohn, D. / Tran, T. / Vissinga, C. / Wannberg, S. / Whittington, D.A. / Whoriskey, J. / Yu, G. / Zalameda, L. / Zhang, X. / Cushing, T.D. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.65 Å |
Structure data | PDB-5kae: |
Chemicals | ChemComp-SO4: ChemComp-6RF: ChemComp-HOH: |
Source |
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Keywords | Transferase/Transferase Inhibitor / phosphotransferase / inhibitor / inflammatory disease / Transferase-Transferase Inhibitor complex |