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-Structure paper
Title | Structure-Based Optimization of HIF-2alpha Agonists That Synergistically Enhance Erythropoietin Production with PHD Inhibitors |
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Journal, issue, pages | J. Med. Chem., Year 2025 |
Publish date | Jan 15, 2025 (structure data deposition date) |
![]() | Wu, D. / Zhuang, J. / Li, F. / Chen, X. / Diao, X. |
![]() | ![]() |
Methods | X-ray diffraction |
Resolution | 2.78 - 3.2 Å |
Structure data | ![]() PDB-9ljx: ![]() PDB-9ljy: ![]() PDB-9loh: ![]() PDB-9loi: |
Chemicals | ![]() PDB-1ekb: ![]() ChemComp-HOH: ![]() PDB-1ej9: ![]() PDB-1ej8: ![]() PDB-1eka: |
Source |
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![]() | TRANSCRIPTION / hypoxia-inducible factor (HIF)-2 / transcriptor |