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-Structure paper
Title | Novel USP7 inhibitors demonstrate potent anti-cancer activity in models of AML, synergy with BCL2 inhibition, and a differentiated mechanism of action |
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Journal, issue, pages | To Be Published |
Publish date | Jun 3, 2022 (structure data deposition date) |
Authors | Futran, A.S. / Lu, T. / Amberg-Johnson, K. / Xu, J. / Yang, X. / He, S. / Boyce, S. / Bell, J. / Pelletier, R. / Suzuki, T. ...Futran, A.S. / Lu, T. / Amberg-Johnson, K. / Xu, J. / Yang, X. / He, S. / Boyce, S. / Bell, J. / Pelletier, R. / Suzuki, T. / Huang, X. / Qian, H. / Fang, L. / Xing, L. / Xu, Z. / Kurtz, S.E. / Tyner, J.W. / Tang, W. / Guo, T. / Akinsanya, K. / Madge, D. / Jensen, K. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.26 Å |
Structure data | PDB-8d4z: |
Chemicals | ChemComp-QBL: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/INHIBITOR / USP7 / ALLOSTERIC / INHIBITOR / HYDROLASE / HYDROLASE-INHIBITOR complex |