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-Structure paper
Title | Mek1 adopts DFG-out conformation when bound to an analog of E6201. |
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Journal, issue, pages | To Be Published |
Publish date | Feb 2, 2016 (structure data deposition date) |
![]() | Larsen, N.A. / Bloudoff, K. / Subramanian, V. / Nomoto, K. / Wang, J. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-5hze: |
Chemicals | ![]() ChemComp-E62: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
Source |
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![]() | Transferase/Transferase Inhibitor / Mek1 / E6201 / Covalent inhibitor / kinase / Mek-1 / MAP2K1 / DFG-out / Transferase-Transferase Inhibitor complex |