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| Title | B-nor-methylene Colchicinoid PT-100 Selectively Induces Apoptosis in Multidrug-Resistant Human Cancer Cells via an Intrinsic Pathway in a Caspase-Independent Manner |
|---|---|
| Journal, issue, pages | Acs Omega, Vol. 7, Page 2591-2603, Year 2022 |
| Publish date | Nov 18, 2019 (structure data deposition date) |
Authors | Stein, A. / Hilken nee Thomopoulou, P. / Frias, C. / Hopff, S.M. / Varela, P. / Wilke, N. / Mariappan, A. / Neudorfl, J.M. / Fedorov, A.Y. / Gopalakrishnan, J. ...Stein, A. / Hilken nee Thomopoulou, P. / Frias, C. / Hopff, S.M. / Varela, P. / Wilke, N. / Mariappan, A. / Neudorfl, J.M. / Fedorov, A.Y. / Gopalakrishnan, J. / Gigant, B. / Prokop, A. / Schmalz, H.G. |
External links | Acs Omega / Search PubMed |
| Methods | X-ray diffraction |
| Resolution | 2.121 Å |
| Structure data | ![]() PDB-6th4: |
| Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-GDP: ![]() ChemComp-N9B: ![]() ChemComp-HOH: |
| Source |
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Keywords | CELL CYCLE / cytoskeleton / cell division / intracellular transport / TRANSPORT PROTEIN / MICROTUBULE |
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