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-Structure paper
Title | Identification and Characterization of a Small Molecule Inhibitor of the Ubiquitin Activating Enzyme (TAK-243) |
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Journal, issue, pages | To be published |
Publish date | Oct 25, 2016 (structure data deposition date) |
![]() | Hyer, M. / Milhollen, M. / Ciavarri, J. / Fleming, P. / Traore, T. / Sappal, D. / Huck, J. / Shi, J. / Gavin, J. / Brownell, J. ...Hyer, M. / Milhollen, M. / Ciavarri, J. / Fleming, P. / Traore, T. / Sappal, D. / Huck, J. / Shi, J. / Gavin, J. / Brownell, J. / Yang, Y. / Stringer, B. / Griffin, R. / Bruzzese, F. / Soucy, T. / Duffy, J. / Rabino, C. / Riceberg, J. / Hoar, K. / Lublinsky, A. / Menon, S. / Sintchak, M. / Bump, N. / Pulukuri, S. / Amidon, B. / Langston, S. / Tirrell, S. / Kuranda, M. / Veiby, P. / Newcomb, J. / Li, P. / Wu, J. / Dick, L. / Greenspan, P. / Galvin, K. / Manfredi, M. / Claibrone, C. / Bence, N. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-5tr4: |
Chemicals | ![]() ChemComp-61T: ![]() ChemComp-HOH: |
Source |
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![]() | LIGASE/LIGASE INHIBITOR / LIGASE-LIGASE INHIBITOR complex |