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-Structure paper
Title | Structural and biophysical insights into the mode of covalent binding of rationally designed potent BMX inhibitors |
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Journal, issue, pages | Chem. Biol., Year 2020 |
Publish date | Nov 22, 2018 (structure data deposition date) |
Authors | Seixas, J.D. / Sousa, B.B. / Marques, M.C. / Guerreiro, A. / Traquete, R. / Rodrigues, T. / Albuquerque, I.S. / Sousa, M.F.Q. / Lemos, A.R. / Sousa, P.M.F. ...Seixas, J.D. / Sousa, B.B. / Marques, M.C. / Guerreiro, A. / Traquete, R. / Rodrigues, T. / Albuquerque, I.S. / Sousa, M.F.Q. / Lemos, A.R. / Sousa, P.M.F. / Bandeiras, T.M. / Wu, D. / Doyle, S.K. / Robinson, C.V. / Koehler, A.N. / Corzana, F. / Matias, P.M. / Bernardes, G.J.L. |
External links | Chem. Biol. / Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.001 Å |
Structure data | PDB-6i99: |
Chemicals | ChemComp-H88: ChemComp-HOH: |
Source |
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Keywords | CYTOSOLIC PROTEIN / Cytoplasmic tyrosine-kinase BMX / Homo Sapiens |