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| Title | c-KIT kinase domain in complex with IDRX-42 via soaking |
|---|---|
| Journal, issue, pages | To Be Published |
| Publish date | Feb 15, 2024 (structure data deposition date) |
Authors | Teuber, A. / Niggenaber, J. / Kleinboelting, S.B. / Landel, I. / Warmuth, J. / Busick, D. / Mueller, M.P. / Bauer, S. / Rauh, D. |
External links | Search PubMed |
| Methods | X-ray diffraction |
| Resolution | 2 Å |
| Structure data | ![]() PDB-8s1b: |
| Chemicals | ![]() ChemComp-K3R: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
| Source |
|
Keywords | TRANSFERASE / stem cell factor receptor / GIST / cancer / inhibitor / resistances |
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