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-Structure paper
Title | Structure-Based Design, Synthesis and Biological Evaluation of Potent and Selective Macrocyclic Chk1 Inhibitors |
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Journal, issue, pages | To be Published |
Publish date | Jan 26, 2007 (structure data deposition date) |
![]() | Tong, Y. / Claiborne, A. / Stewart, K.D. / Park, C. / Kovar, P. / Chen, Z. / Credo, R.B. / Gwaltney, S.L. / Zhang, H. / Rosenberg, S.H. ...Tong, Y. / Claiborne, A. / Stewart, K.D. / Park, C. / Kovar, P. / Chen, Z. / Credo, R.B. / Gwaltney, S.L. / Zhang, H. / Rosenberg, S.H. / Sham, H.L. / Sowin, T.J. / Lin, N.H. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.6 Å |
Structure data | ![]() PDB-2e9p: |
Chemicals | ![]() ChemComp-77A: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / Protein-inhibitor Complex |